Methyltestosterone tablets or capsules

What is this medication?

METHYLTESTOSTERONE (meth uhl tes TOS ter one) is a male hormone. This medicine is used to treat low testosterone levels in males. It is also used to treat certain breast cancers in women.

This medicine may be used for other purposes; ask your health care provider or pharmacist if you have questions.

COMMON BRAND NAME(S): Android, Methitest, Testred, Virilon

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What should I tell my care team before I take this medication?

They need to know if you have any of these conditions:

  • Diabetes
  • Prostate cancer
  • Prostate problems
  • Other medical condition
  • An unusual or allergic reaction to methyltestosterone, other medications, foods, dyes, or preservatives
  • Pregnant or trying to get pregnant
  • Breast-feeding

How should I use this medication?

Take this medication by mouth with a glass of water. Follow the directions on the prescription label. Take your doses at regular intervals. Do not take your medication more often than directed.

Talk to your care team about the use of this medication in children. This medication is not approved for use in children.

Overdosage: If you think you have taken too much of this medicine contact a poison control center or emergency room at once.

NOTE: This medicine is only for you. Do not share this medicine with others.

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What if I miss a dose?

If you miss a dose, take it as soon as you can. If it is almost time for your next dose, take only that dose. Do not take double or extra doses.

What may interact with this medication?

  • Medications for diabetes
  • Oxyphenbutazone
  • Warfarin

This list may not describe all possible interactions. Give your health care provider a list of all the medicines, herbs, non-prescription drugs, or dietary supplements you use. Also tell them if you smoke, drink alcohol, or use illegal drugs. Some items may interact with your medicine.

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What should I watch for while using this medication?

Visit your care team for regular check-ups. You will need to have important blood work done while you are taking this medication.

This medication may lower blood sugar in patients with diabetes. If you have diabetes, monitor your blood sugar and report any changes.

This medication is banned from use in athletes by the US and the International Olympic Committees and other athletic organizations.

What side effects may I notice from receiving this medication?

Side effects that you should report to your doctor or health care professional as soon as possible:

  • allergic reactions like skin rash, itching or hives, swelling of the face, lips, or tongue
  • breast enlargement
  • breathing problems
  • changes in mood, especially anger, depression, or rage
  • dark urine
  • in women: acne, change in monthly cycle, deep voice, enlarged clitoris, more face hair
  • nausea, vomiting
  • stomach pain
  • swelling of the ankles or legs
  • too frequent or persistent erections
  • trouble passing urine
  • unusual bleeding or bruising
  • yellowing of eyes, skin

Side effects that usually do not require medical attention (report to your doctor or health care professional if they continue or are bothersome):

  • acne in men
  • change in sex drive or performance
  • headache

This list may not describe all possible side effects. Call your doctor for medical advice about side effects. You may report side effects to FDA at 1-800-FDA-1088.

Where should I keep my medication?

Keep out of the reach of children and pets. This medication can be abused. Keep your medication in a safe place to protect it from theft. Do not share this medication with anyone. Selling or giving away this medication is dangerous and against the law.

Store at room temperature between 15 and 30 degrees C (59 and 86 degrees F). Throw away any unused medication after the expiration date.

NOTE: This sheet is a summary. It may not cover all possible information. If you have questions about this medicine, talk to your doctor, pharmacist, or health care provider.

Copyright ©2024 Elsevier Inc. All Rights Reserved.

Terms of use.

Note: Introduction and Additional Common Questions written and medically approved by Cleveland Clinic professionals.

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